


- Yuntong Zhai, Xiaofei Chen, Wei Zhou, Mengyang Fan, Yisheng Lai, and Dawei Ma*, Pd-Catalyzed dimethylation of tyrosine-derived picolinamide for synthesis of (S)-N-boc-2,6-dimethyltyrosine and its analogues Copper-Catalyzed Diaryl Ether Formation from (Hetero)aryl Halides at Low Catalytic Loadings. J. Org. Chem., 2017, 82, 4964−4969.
- Xiangbo Zhao, Wu Li, Junjie Wang, Dawei Ma*, Convergent route to ent-Kaurane diterpenoids: Total Ssynthesis of Lungshengenin D and 1,6-Diacetoxy-ent-kaura- 9(11),16-dien-12,15-dione. J. Am. Chem. Soc., 2017, 139(8), 2932-2935.

- Xuning Wang, Songtao Niu, Lanting Xu, Chao Zhang, Lingxing Meng, Xiaojing Zhang,* and Dawei Ma*, Pd-Catalyzed dimethylation of tyrosine-derived picolinamide for synthesis of (S)-N-boc-2,6-dimethyltyrosine and its analogues. Org. Lett., 2017, 19(1), 246-249.
- Subhadip De, Junli Yin, and Dawei Ma* Copper-Catalyzed Coupling Reaction of (Hetero)Aryl Chlorides and Amides. Org. Lett. 2017, 19, 4864−4867.
- Subhajit Bhunia, Govind Goroba Pawar, S. Vijay Kumar, Yongwen Jiang and Dawei Ma* Selected Copper-Based Reactions for C-N, C-O, C-S and C-C Bond Formation. Angew. Chem. Int. Ed. 2017, 56, 16136–16179.

- Songtao Niu, Jinlong Zhao, Xi Jiang, Yongwen Jiang, Xiaojing Zhang, Tiemin Sun and Dawei Ma* A New Class of Amide Ligands Enable Cu-Catalyzed Coupling of Sodium Methanesulfinate with (Hetero)aryl Chlorides. Chin. J. Chem. 2017, 35, 1661—1664.
- Subhajit Bhunia, S. Vijay Kumar, and Dawei Ma* N,N’- Bisoxalamides Enhance the Catalytic Activity in Cu-Catalyzed Coupling of (Hetero)Aryl Bromides with Anilines and Secondary Amines. J. Org. Chem. 2017, 82, 12603−12612.
- Shanghua Xia, Lu Gan, Kailiang Wang, Zheng Li, Dawei Ma “Copper-Catalyzed Hydroxylation of (Hetero)aryl Halides under Mild Conditions” Journal of the American Chemical Society 2016, 138(19), 13493-13496

- Lanting Xu, Lushi Tan, Dawei Ma “Iridium(III)-Catalyzed Regioselective C7-Amination of N-Pivaloylindoles with Sulfonoazides” Journal of Organic Chemistry 2016, 81(21), 10476-10483.
- Mengyang Fan, Wei Zhou, Yongwen Jiang, Dawei Ma* ‘CuI/Oxalamide Catalyzed Couplings of (Hetero)aryl Chlorides and Phenols for Diaryl Ether Formation’ Angewandte Chemie, International Edition 2016, 55(21), 6211-6215.








- Junshan Tian, Jiankang Zhong, Yunsheng Li, and Dawei Ma*, Organocatalytic and Scalable Synthesis of the Anti-Influenza Drugs Zanamivir, Laninamivir, and CS-8958. Angewandte Chemie, International Edition, 2014, 53, 13885-13888.
- Mingxing Teng, Weiwei Zi, and Dawei Ma*, Total Synthesis of the Monoterpenoid Indole Alkaloid (±)-Aspidophylline A. Angewandte Chemie, International Edition, 2014, 53, 1814-11817.
- Chengang Zhou and Dawei Ma*, A copper-catalyzed coupling reaction of vinyl halides and carbazates: application in the assembly of polysubstituted pyrroles, Chemical Communications, 2014, 50, 3085-3088.
- Huan Liu, Guangde Jiang, Xixian Pan, Xiaolong Wan, Yisheng Lai, Dawei Ma*, and Weiqing Xie, Highly Asymmetric Bromocyclization of Tryptophol: Unexpected Accelerating Effect of DABCO-Derived Bromine Complex, Organic Letters 2014, 16, 1908-1911.
- Wu, Mingyao; Ma, Dawei *Total Syntheses of (±)-Spiroquinazoline, (-)-Alantryphenone, (+)-Lapatin A, and (-)-Quinadoline B. Angewandte Chemie, International Edition 2013, 52, 9759-9762.
- Xie Weiqing; Jiang Guangde; Liu Huan; Hu Jiadong; Pan Xixian; Zhang Hui; Wan Xiaolong; Lai Yisheng; Ma Dawei* Highly Enantioselective Bromocyclization of Tryptamines and Its Application in the Synthesis of (-)-Chimonanthine. Angewandte Chemie, International edition 2013, 52, 12924-12927.
- Wei, Yi; Zhao, Duo; Ma, Dawei *Total Synthesis of the Indole Alkaloid (±)- and (+)-Methyl N-Decarbomethoxychanofruticosinate. Angewandte Chemie, International Edition, 2013, 52, 12988-12991.
- Fan, Mengyang; Ma, Dawei *Palladium-Catalyzed Direct Functionalization of 2-Aminobutanoic Acid Derivatives: Application of a Convenient and Versatile Auxiliary. Angewandte Chemie, International Edition 2013, 52(46), 12152-12155
- Xie, Weiqing; Zuo, Zhiwei; Zi, Weiwei; Ma, Dawei* Intramolecular oxidative coupling: applications in synthesis of complex indole akaloid scaffolds Youji Huaxue 2013, 33(5), 869-876.
- Jiang, Yongwen; Xu, Lanting; Zhou, Chenggang; Ma, Dawei* Cu-catalyzed Ullmann-type C-heteroatom bond formation: the key role of dinucleating ancillary ligands RSC Catalysis Series 2013, 11(C-H and C-X Bond Functionalization), 1-45.
- Chen, Yu; Lu, Yuwei; Zou, Qing; Chen, Huansheng; Ma, Dawei* A Scalable Process to the Key Intermediate of Cilazapril, (S)-1-Benzyloxycarbonylhexahydropyridazine-3-carboxylic Acid, Through a Novel Cascade Course Organic Process Research & Development 2013, 17(9), 1209-1213.
- Xie, Weiqing; Wang, Hexiang; Fan, Feng; Tian, Junshan; Zuo, Zhiwei; Zi, Weiwei; Gao, Kun; Ma, Dawei* Diastereoselective construction of continuous all-carbon quaternary centers via intramolecular oxidative coupling reaction Tetrahedron Letters 2013, 54(33), 4392-4396.
- Kishor, Chandan; Arya, Tarun; Reddi, Ravikumar; Chen, Xiaochun; Saddanapu, Venkateshwarlu; Marapaka, Anil Kumar; Gumpena, Rajesh; Ma, Dawei*; Liu, Jun O.; Addlagatta, Anthony Identification, Biochemical and Structural Evaluation of Species-Specific Inhibitors against Type I Methionine Aminopeptidases Journal of Medicinal Chemistry 2013, 56(13), 5295-5305.
- Xie, Siwei; Qin, Peng; Li, Meng; Zhang, Xiaojing; Jiang, Yongwen; Ma, Dawei* Synthesis of 2-alkyl-2-arylcyanoacetates via CuI/sodium picolinate-catalyzed direct arylation of a-substituted cyanoacetates Tetrahedron Letters 2013, 54(29), 3889-3891.
- Yin, Hongfei; Chen, Bing; Zhang, Xiaojing; Yang, Xinye; Zhang, Yihua; Jiang, Yongwen; Ma, Dawei* Assembly of N,N-disubstituted-N'-arylureas via a copper-catalyzed one-pot three-component reaction of aryl bromides, potassium cyanate, and secondary amines Tetrahedron 2013, 69(26), 5326-5330.
- Zhang, Pengtao; Yang, Xinye; Zhang, Feiran; Gabelli, Sandra B.; Wang, Renxiao; Zhang, Yihua; Bhat, Shridhar; Chen, Xiaochun; Furlani, Manuel; Amzel, L. Mario; et al Pyridinylpyrimidines selectively inhibit human methionine aminopeptidase-1 Bioorganic & Medicinal Chemistry 2013, 21(9), 2600-2617.
- Xu, Lanting; Peng, Yinsheng; Pan, Qiangbiao; Jiang, Yongwen; Ma, Dawei *Assembly of Substituted 3-Aminoindazoles from 2-Bromobenzonitrile via a CuBr-Catalyzed Coupling/Condensation Cascade Process Journal of Organic Chemistry 2013, 78(7), 3400-3404.
- Zhang, Ye; Xing, Hui; Xie, Weiqing; Wan, Xiaolong; Lai, Yisheng; Ma, Dawei* Asymmetric, Regioselective Bromohydroxylation of 2-Aryl-2-propen-1-ols Catalyzed by Quinine-Derived Catalysts Advanced Synthesis & Catalysis 2013, 355, 68-72.
- Zhang, Feiran; Bhat, Shridhar; Gabelli, Sandra B.; Chen, Xiaochun; Miller, Michelle S.; Nacev, Benjamin A.; Cheng, Yim Ling; Meyers, David J.; Tenney, Karen; Shim, Joong Sup; Crews, Phillip; Amzel, L. Mario; Ma, Dawei*; Liu, Jun O. Pyridinylquinazolines Selectively Inhibit Human Methionine Aminopeptidase-1 in Cells Journal of Medicinal Chemistry 2013, 56, 3996-4016.
- Songchuan Tian, Weiwei Zi, Dawei Ma* ‘Potentially Biomimetic Total Synthesis and Relative Stereochemical Assignment of (±)-Gracilamine’ Angewandte Chemie, International Edition 2012, 51(40), 10141-10144
- Fan, Feng; Xie, Weiqing; Ma, Dawei* Cascade annulation of malonic diamides: a concise synthesis of polycyclic pyrroloindolines, Chemical Communications (Cambridge, United Kingdom) 2012, 48, 7571-7573.
- Fan, Feng; Xie, Weiqing; Ma, Dawei* Construction of Polycyclic Spiro-indolines via an Intramolecular Oxidative Coupling/Cyclization Cascade Reaction Process, Organic Letters 2012, 14, 1405-1407.
- Huo, Lele; Ma, Anqi; Zhang, Yihua; Ma, Dawei* Assembly of 4-Substituted 3-Nitro-1,2,3,4-tetrahydropyridines via Organocatalytic Michael Addition, Advanced Synthesis & Catalysis 2012, 354, 991-994.
- Li, Jiaojiao; Zhang, Yihua; Jiang, Yongwen; Ma, Dawei* CuI/N,N-dimethylglycine-catalyzed synthesis of N-aryloxazolidinones from aryl bromides, Tetrahedron Letters 2012, 53, 3981-3983.
- Li, Jiaojiao; Zhang, Yihua; Jiang, Yongwen; Ma, Dawei* CuI-catalyzed one-pot synthesis of benzothiazolones from 2-iodoanilines-derived carbamates and sodium sulfide, Tetrahedron Letters 2012, 53, 2511-2513.
- Liu, Qing; Li, Na; Yuan, Yunyun; Lu, Huili; Wu, Xiaoyan; Zhou, Caihong; He, Min; Su, Haoran; Zhang, Meng; Wang, Jia; Wang, Bao; Wang, You; Ma, Dawei*; Ye, Yang; Weiss, Hans-Christoph; Gesing Ernst, R. F.; Liao, Jiayu; Wang, Ming-Wei Cyclobutane derivatives as novel nonpeptidic small molecule agonists of glucagon-like peptide-1 receptor, J Med Chem 2012, 55, 250-267.
- Wang, Leilei; Zhang, Xiaojing; Ma, Dawei* Organocatalytic Michael addition of aldehydes to trisubstituted nitroolefins, Tetrahedron 2012, 68, 7675-7679.
- Xing, Hui; Zhang, Ye; Lai, Yisheng; Jiang, Yongwen; Ma, Dawei* Synthesis of Symmetrical and Unsymmetrical N,N'-Diaryl Guanidines via Copper/N-Methylglycine-Catalyzed Arylation of Guanidine Nitrate, Journal of Organic Chemistry 2012, 77, 5449-5453.
- Xiong, Xiaodong; Jiang, Yongwen; Ma, Dawei* Assembly of N,N-Disubstituted Hydrazines and 1-Aryl-1H-indazoles via Copper-Catalyzed Coupling Reactions, Organic Letters 2012, 14, 2552-2555.
- Xu, Lanting; Jiang, Yongwen; Ma, Dawei* Synthesis of 3-Substituted and 2,3-Disubstituted Quinazolinones via Cu-Catalyzed Aryl Amidation, Organic Letters 2012, 14, 1150-1153.
- Yang, Xinye; Xing, Hui; Zhang, Ye; Lai, Yisheng; Zhang, Yihua; Jiang, Yongwen; Ma, Dawei* CuI/8-Hydroxyquinaldine Promoted N-Arylation of Indole and Azoles, Chinese Journal of Chemistry 2012, 30, 875-880.
- Zhang, Yu; Yang, Xinye; Yao, Qizheng; Ma, Dawei* CuI/DMPAO-Catalyzed N-Arylation of Acyclic Secondary Amines, Organic Letters 2012, 14, 3056-3059.
- Zi, Weiwei; Xie, Weiqing; Ma, Dawei* Total Synthesis of Akuammiline Alkaloid (-)-Vincorine via Intramolecular Oxidative Coupling, Journal of the American Chemical Society 2012, 134, 9126-9129.
- Chen, Gang; Xia, Hongguang; Cai, Yu; Ma, Dawei*; Yuan, Junying; Yuan, Chengye Diphenylbutylpiperidine-based cell autophagy inducers: Design, synthesis and SAR studies, MedChemComm 2011, 2, 315-320.
- Chen, Gang; Xia, Hongguang; Cai, Yu; Ma, Dawei*; Yuan, Junying; Yuan, Chengye Synthesis and SAR study of diphenylbutylpiperidines as cell autophagy inducers, Bioorganic & Medicinal Chemistry Letters 2011, 21, 234-239.
- Han, Shuai; Pan, Heling; Zhang, Jianhua; Tan, Li; Ma, Dawei*; Yuan, Junying; Wu, Jia-Rui Identification of a small molecule activator of novel PKCs for promoting glucose-dependent insulin secretion, Cell Research 2011, 21, 588-599.
- Li, Wenhua; Yu, Shouyun; Jin, Mingzhi; Xia, Hongguang; Ma, Dawei* Total synthesis and cytotoxicity of bisebromoamide and its analogues, Tetrahedron Letters 2011, 52, 2124-2127.
- Liu, Junli; Xia, Hongguang; Kim, Minsu; Xu, Lihua; Li, Ying; Zhang, Lihong; Cai, Yu; Norberg, Helin Vakifahmetoglu; Zhang, Tao; Furuya, Tsuyoshi; Jin, Minzhi; Zhu, Zhimin; Wang, Huanchen; Yu, Jia; Li, Yanxia; Hao, Yan; Choi, Augustine; Ke, Hengming; Ma, Dawei*; Yuan, Junying Beclin1 Controls the Levels of p53 by Regulating the Deubiquitination Activity of USP10 and USP13, Cell (Cambridge, MA, United States) 2011, 147, 223-234.
- Ma, Dawei*; Jiang, Yongwen Cu(I)/amino acid catalyzed coupling reactions of aryl halides and nucleophiles: applications in large-scale production, Chimia 2011, 65, 914-918.
- Ma, Dawei*; Lu, Xu; Shi, Liu; Zhang, Hui; Jiang, Yongwen; Liu, Xiangqian Domino condensation/S-arylation/heterocyclization reactions: copper-catalyzed three-component synthesis of 2-N-substituted benzothiazoles, Angewandte Chemie, International Edition 2011, 50, 1118-1121.
- Shi, Liu; Liu, Xiangqian; Zhang, Hui; Jiang, Yongwen; Ma, Dawei* Synthesis of 2-thio-substituted benzothiazoles via a domino condensation/S-arylation/heterocyclization process, Journal of Organic Chemistry 2011, 76, 4200-4204.
- Sun, Xuefeng; Ma, Dawei* Organocatalytic Approach for the Syntheses of Corynantheidol, Dihydrocorynantheol, Protoemetinol, Protoemetine, and Mitragynine, Chemistry--An Asian Journal, 2011, 6, 2158-2165.
- Wang, You; Zhu, Shaolin; Ma, Dawei* Organocatalytic Approach to Polysubstituted Piperidines and Tetrahydropyrans, Organic Letters 2011, 13, 1602-1605.
- Yu, Shouyun; Zhu, Shaolin; Pan, Xianhua; Yang, Jiade; Ma, Dawei* Reinvestigation on total synthesis of kaitocephalin and its isomers, Tetrahedron 2011, 67, 1673-1680.
- Chang M., Kanwar N., Feng E., Siu A., Liu X., Ma D., Jongstra J., PIM kinase inhibitors downregulate STAT3Tyr705 phosphorylation. Mol. Cancer Ther. 2010, 9,2478.
- Ben, Li; Jones, Eric Dale; Zhou, Enkun; Li, Chen; Baylis, Dean Cameron; Yu, Shanghai; Wang, Miao; He, Xing; Coates, Jonathan Alan Victor; Rhodes, David Ian; Pei, Gang; Deadman, John Joseph; Xie, Xin; Ma, Dawei Studies on the structure-activity relationship of 1,3,3,4-tetra-substituted pyrrolidine embodied CCR5 receptor antagonists. Part 1: Tuning the N-substituents, Bioorganic & Medicinal Chemistry Letters 2010, 20, 4012-4014.
- Hao, Chao; Zhang, Yihua; Jiang, Yongwen; Ma, Dawei* CuBr/N,N-dimethylglycine-catalyzed coupling reaction of 2-chlorotrifluoroacetanilides with phenols at mild conditions, Chinese Journal of Chemistry 2010, 28, 1645-1650.
- Li, Ben; Jones, Eric Dale; Zhou, Enkun; Chen, Li; Baylis, Dean Cameron; Yu, Shanghai; Wang, Miao; He, Xing; Coates, Jonathan Alan Victor; Rhodes, David Ian; Pei, Gang; Deadman, John Joseph; Xie, Xin; Ma, Dawei* Studies on the structure-activity relationship of 1,3,3,4-tetra-substituted pyrrolidine embodied CCR5 receptor antagonists. Part 2: Discovery of highly potent anti-HIV agents, Bioorganic & Medicinal Chemistry Letters 2010, 20, 5334-5336.
- Li, Wenhua; Schlecker, Andreas; Ma, Dawei* Total synthesis of antimicrobial and antitumor cyclic depsipeptides, Chemical Communications (Cambridge, United Kingdom) 2010, 46, 5403-5420.
- Lu, Xu; Shi, Liu; Zhang, Hui; Jiang, Yongwen; Ma, Dawei* Assembly of N-substituted pyrrolo[2,1-c][1,4]benzodiazepine-5,11-diones via copper catalyzed aryl amination, Tetrahedron 2010, 66, 5714-5718.
- Ma, Anqi; Ma, Dawei* Enantioselective Synthesis of Polysubstituted Cyclopentanones by Organocatalytic Double Michael Addition Reactions, Organic Letters 2010, 12, 3634-3637.
- Ma, Dawei*; Geng, Qian; Zhang, Hui; Jiang, Yongwen Assembly of Substituted Phenothiazines by a Sequentially Controlled CuI/L-Proline-Catalyzed Cascade C-S and C-N Bond Formation, Angewandte Chemie, International Edition 2010, 49, 1291-1294.
- Maurer, Stefan; Liu, Wei; Zhang, Xiaojing; Jiang, Yongwen; Ma, Dawei* An efficient synthesis of phenol via CuI/8-hydroxyquinoline-catalyzed hydroxylation of aryl halides and potassium hydroxide, Synlett 2010, 976-978.
- Wang, You; Xu, Lanting; Ma, Dawei* CuI/L-Proline-Catalyzed Coupling of Substituted 3-Iodoprop-2-en-1-ols with 1-Alkynes and Subsequent Cyclization: A Convenient Approach for Synthesizing Polysubstituted Furans, Chemistry--An Asian Journal 2010, 5, 74-76.
- Xia, Hong-guang; Zhang, Lihong; Chen, Gang; Zhang, Tao; Liu, Junli; Jin, Mingzhi; Ma, Xiuquan; Ma, Dawei*; Yuan, Junying Control of basal autophagy by calpain1 mediated cleavage of ATG5, Autophagy 2010, 6, 61-66.
- Xu, Danhua; Zhang, Yihua; Ma, Dawei* Organocatalytic approach to 3,5,6-trisubstituted and 4,6-disubstituted tetrahydropyran-2-ones, Tetrahedron Letters 2010, 51, 3827-3829.
- Xu, Lanting; Jiang, Yongwen; Ma, Dawei* Synthesis of tetrahydropyrrolo[1,2-a]quinoxalines and tetrahydropyrido[1,2-a]quinoxalines via a one-pot CuI-catalyzed aryl amination-hydrolysis-condensation process, Synlett, 2010, 2285-2288.
- Zhou, Qianghui; Chen, Xiaofei; Ma, Dawei Asymmetric, Protecting-Group-Free Total Synthesis of (-)-Englerin A, Angewandte Chemie, International Edition 2010, 49, 3513-3516.
- Zhu, Shaolin; Yu, Shouyun; Wang, You; Ma, Dawei* Organocatalytic Michael addition of aldehydes to protected 2-amino-1-nitroethenes: the practical syntheses of oseltamivir (Tamiflu) and substituted 3-aminopyrrolidines, Angewandte Chemie, International Edition 2010, 49, 4656-4660.
- Zi, Weiwei; Yu, Shouyun; Ma, Dawei* A Convergent Route to the Galbulimima Alkaloids (-)-GB 13 and (+)-GB 16, Angewandte Chemie, International Edition 2010, 49, 5887-5890.
- Zi, Weiwei; Yu, Shouyun; Ma, Dawei* Synthetic Studies toward Galbulimima Alkaloid (-)-GB 13 and (+)-GB 16 and (-)-Himgaline, Chemistry, an Asian journal 2010,6,573.
- Zuo, Zhiwei; Xie, Weiqing; Ma, Dawei* Total Synthesis and Absolute Stereochemical Assignment of (-)-Communesin F, Journal of the American Chemical Society 2010, 132, 13226-13228.
发表时间:2015-03-01 阅读次数:2652次